SCHEMBL6814839

SCHEMBL6814839

COc1ccc(-c2ncnc(NCCC3CC3)c2N)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 5/20 0.39
ENPP1 P22413 1/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
CRHR2 Q13324 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDC7 O00311 1/20 0.35
CCNT1 O60563 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CSNK1D P48730 1/20 0.35
CDK9 P50750 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
DBF4 Q9UBU7 1/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821870 0.96 ENPP1 (0.36) CRHR1ENPP1HSP90AA1HSP90AB1CRHR2
SCHEMBL6818769 0.88 FFAR4 (0.35) CRHR1CCNT1JAK2JAK1
SCHEMBL6813739 0.85 DYRK1A (0.38) CRHR1ENPP1DYRK1AJAK2JAK1
SCHEMBL6817533 0.79 HSP90AA1 (0.37) CRHR1HSP90AA1HSP90AB1CRHR2CDC7
SCHEMBL6082630 0.78 IDH2 (0.42) CRHR1HSP90AA1HSP90AB1DYRK1ACDC7
SCHEMBL6082635 0.78 IDH2 (0.42) CRHR1HSP90AA1HSP90AB1DYRK1ACDC7
SCHEMBL6082839 0.76 IDH2 (0.39) CRHR1HSP90AA1HSP90AB1DYRK1ACDC7
SCHEMBL6082842 0.76 IDH2 (0.39) CRHR1HSP90AA1HSP90AB1DYRK1ACDC7
SCHEMBL6818798 0.76 ABL1 (0.36) CRHR1KDRJAK2JAK1JAK3
SCHEMBL6818015 0.76 ACP1 (0.36) CRHR1HSP90AA1HSP90AB1CRHR2CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed