SCHEMBL6817320

SCHEMBL6817320

Cc1c(OCCN(C)C)c2ccc(Cl)cc2n1Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
RAD52 P43351 1/20 0.45
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 1/20 0.44
S1PR3 Q99500 1/20 0.41
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
PLA2G2A P14555 3/20 0.40
KDM4E B2RXH2 2/20 0.40
LTA4H P09960 1/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
GUCY1B2 O75343 1/20 0.39
CYP1A2 P05177 1/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821061 0.91 TDP1 (0.53) TDP1MEN1GAAMAPTRAD52
SCHEMBL6817497 0.87 TDP1 (0.52) TDP1MEN1GAAMAPTRAD52
SCHEMBL6817304 0.86 ESR1 (0.43) TDP1S1PR3MAPK8MAPK9KDM4E
SCHEMBL6820282 0.81 TDP1 (0.42) TDP1MEN1GAAMAPTRAD52
SCHEMBL6821006 0.81 TDP1 (0.52) TDP1MEN1GAAMAPTRAD52
SCHEMBL6820985 0.80 KMT2A (0.56) TDP1MEN1GAAMAPTRAD52
SCHEMBL6820713 0.79 TDP1 (0.41) TDP1MEN1GAAMAPTRAD52
SCHEMBL3928794 0.78 HTR6 (0.50) KDM4EHTR1ADRD3HTR6
SCHEMBL6820242 0.78 KDM4E (0.45) TDP1GAAALDH1A1KDM4E
SCHEMBL6917019 0.77 ESR1 (0.48) TDP1MEN1GAAMAPTRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048331-A1 N-ARYLALKYL-3-AMINOALKOXYINDOLES AND THEIR USE AS 5-HT LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2004-06-10 WO claimed
WO-2004048331-A1 N-ARYLALKYL-3-AMINOALKOXYINDOLES AND THEIR USE AS 5-HT LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2004-06-10 WO disclosed