SCHEMBL6817877

SCHEMBL6817877

O=C(O)c1cc(Br)ccc1NC(=O)c1onc2cc(Cl)ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.46
ACLY P53396 1/20 0.46
DNMT3A Q9Y6K1 1/20 0.46
SORT1 Q99523 1/20 0.46
AKR1C2 P52895 3/20 0.46
AKR1C1 Q04828 3/20 0.46
AKR1C4 P17516 2/20 0.46
AKR1C3 P42330 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
METAP2 P50579 1/20 0.45
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KCNH2 Q12809 1/20 0.43
SERPINE1 P05121 3/20 0.43
STING1 Q86WV6 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6814011 0.86 ACLY (0.38) GRIK1ACLYDNMT3ASORT1AKR1C2
SCHEMBL6818060 0.85 AKR1C2 (0.51) SORT1AKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL6818553 0.85 AKR1C2 (0.50) ACLYAKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL6818795 0.84 CA12 (0.43) AKR1C2AKR1C1AKR1C4AKR1C3MEN1
SCHEMBL6833190 0.83 HIF1A (0.47) GRIK1ACLYDNMT3ASORT1AKR1C2
SCHEMBL6818370 0.79 METAP2 (0.44) ACLYAKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL6814346 0.75 ALB (0.42) ACLYAKR1C2AKR1C1AKR1C4AKR1C3
SCHEMBL1307332 0.74 PPARG (0.71) GRIK1ACLYDNMT3ASORT1AKR1C2
SCHEMBL6819170 0.74 MEN1 (0.44) AKR1C2AKR1C1AKR1C4AKR1C3MEN1
SCHEMBL1307201 0.74 KCNK2 (0.64) GRIK1ACLYDNMT3AAKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018428-A1 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO disclosed