SCHEMBL6818697

SCHEMBL6818697

O=C(NCc1ccncc1)c1nc2c(o1)CN(Cc1ccccc1)C=N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.44
ROCK2 O75116 1/20 0.44
RPS6KA5 O75582 1/20 0.44
MAP4K4 O95819 1/20 0.44
PRKCG P05129 1/20 0.44
PRKACA P17612 1/20 0.44
RPS6KB1 P23443 1/20 0.44
AKT1 P31749 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
PRKX P51817 1/20 0.44
PRKCD Q05655 1/20 0.44
PRKG2 Q13237 1/20 0.44
ROCK1 Q13464 1/20 0.44
DYRK1A Q13627 1/20 0.44
PRKG1 Q13976 1/20 0.44
PKN2 Q16513 1/20 0.44
CDC42BPA Q5VT25 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
SGK2 Q9HBY8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6818703 0.83 CCNC (0.36) CYP2D6CYP2C9CYP2C19CYP3A4KMT2A
SCHEMBL6704157 0.81 NR4A2 (0.35) CYP2D6CYP2C9CYP2C19GAAKMT2A
SCHEMBL6818691 0.80 CCNC (0.40) CYP2D6CYP2C9CYP2C19CYP3A4CDC7
SCHEMBL6702617 0.76 MMP13 (0.41) MAPK1ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6819957 0.75 NPC1 (0.46) MAPK1ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6819967 0.72 MMP13 (0.39) MAPK1ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6819953 0.72 MMP13 (0.38) MAPK1ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6700620 0.69 MMP13 (0.44) MAPK1ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6289016 0.66 SCD (0.43) ALDH1A1CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL6698728 0.66 PTGER4 (0.47) ALDH1A1MMP13SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed