SCHEMBL6818703

SCHEMBL6818703

NCc1ccncc1.O=C(O)c1nc2c(o1)CN(Cc1ccccc1)C=N2

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
SIGMAR1 Q99720 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
TSHR P16473 2/20 0.32
KDM4E B2RXH2 2/20 0.32
CYP3A4 P08684 3/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C19 P33261 1/20 0.32
CXCR2 P25025 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
PARP1 P09874 1/20 0.31
CES1 P23141 2/20 0.30
FAAH O00519 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP46A1 Q9Y6A2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6704157 0.89 NR4A2 (0.35) CCNCCDK8TSHRCYP2D6CYP2C19
SCHEMBL6818691 0.89 CCNC (0.40) CCNCCDK8TSHRCYP3A4CYP2D6
SCHEMBL6818697 0.83 MAPK1 (0.44) CYP3A4CYP2D6CYP2C19CYP2C9KMT2A
SCHEMBL6822414 0.75 PTGDR2 (0.36) LOXL2TSHR
SCHEMBL6819967 0.68 MMP13 (0.39)
SCHEMBL6292192 0.67 NR4A2 (0.39) TSHRKDM4ECYP2C9MEN1KMT2A
SCHEMBL6822412 0.65 LMNA (0.37) CCNCCDK8TSHR
Isonicotinic Acid SCHEMBL9986818 0.63 NAPRT (0.63) LOXL2TSHRKDM4ECYP3A4CYP2D6
Carbamic Acid SCHEMBL31175940 0.61 LOXL2 (0.73) LOXL2TSHRKDM4ECYP3A4CYP2D6
Acetic Acid SCHEMBL28099257 0.60 LOXL2 (0.70) LOXL2TSHRKDM4ECYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed