SCHEMBL6819957

SCHEMBL6819957

O=C(NCc1ccncc1)c1ccc(CN2C=Nc3oc(C(=O)NCc4ccncc4)nc3C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MMP13 P45452 4/20 0.43
ROCK2 O75116 1/20 0.43
RPS6KA5 O75582 1/20 0.43
MAP4K4 O95819 1/20 0.43
PRKCG P05129 1/20 0.43
PRKACA P17612 1/20 0.43
RPS6KB1 P23443 1/20 0.43
MAPK1 P28482 1/20 0.43
AKT1 P31749 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
PRKX P51817 1/20 0.43
PRKCD Q05655 1/20 0.43
PRKG2 Q13237 1/20 0.43
ROCK1 Q13464 1/20 0.43
DYRK1A Q13627 1/20 0.43
PRKG1 Q13976 1/20 0.43
PKN2 Q16513 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6702617 0.94 MMP13 (0.41) NPC1RAB9AMMP13ROCK2RPS6KA5
SCHEMBL6822413 0.91 L3MBTL1 (0.46) ROCK2ROCK1CYP3A4MAPK14ALDH1A1
SCHEMBL6819967 0.90 MMP13 (0.39) NPC1RAB9AMMP13ROCK2RPS6KA5
SCHEMBL6819953 0.89 MMP13 (0.38) NPC1RAB9AMMP13ROCK2RPS6KA5
SCHEMBL6700620 0.76 MMP13 (0.44) MMP13ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6818697 0.75 MAPK1 (0.44) MMP13ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL6822414 0.74 PTGDR2 (0.36) MMP13LMNASMN1; SMN2HTTMMP2
SCHEMBL6698728 0.67 PTGER4 (0.47) MMP13ALDH1A1SMN1; SMN2HPGD
SCHEMBL6702248 0.67 MMP13 (0.43) MMP13ROCK2RPS6KA5MAP4K4PRKCG
SCHEMBL1569157 0.67 L3MBTL1 (0.77) MMP13ROCK2RPS6KA5MAP4K4PRKCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed