SCHEMBL6819953

SCHEMBL6819953

NC(=O)c1ccncc1.O=C(O)c1ccc(CN2C=Nc3oc(C(=O)NCc4ccncc4)nc3C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 0.38
NAMPT P43490 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PTGER4 P35408 5/20 0.37
PARP1 P09874 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
ROCK2 O75116 1/20 0.36
RPS6KA5 O75582 1/20 0.36
MAP4K4 O95819 1/20 0.36
PRKCG P05129 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KB1 P23443 1/20 0.36
MAPK1 P28482 1/20 0.36
AKT1 P31749 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
PRKX P51817 1/20 0.36
PRKCD Q05655 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6702617 0.95 MMP13 (0.41) MMP13NAMPTNPC1RAB9APTGER4
SCHEMBL6819967 0.92 MMP13 (0.39) MMP13NAMPTNPC1RAB9APTGER4
SCHEMBL6819957 0.89 NPC1 (0.46) MMP13NAMPTNPC1RAB9AALDH1A1
SCHEMBL6822413 0.85 L3MBTL1 (0.46) NAMPTALDH1A1HSD17B10ROCK2ROCK1
SCHEMBL6822412 0.82 LMNA (0.37) NPC1RAB9A
SCHEMBL6698006 0.81 MMP13 (0.49) MMP13PTGER4GSK3B
SCHEMBL6700620 0.78 MMP13 (0.44) MMP13NAMPTPTGER4ALDH1A1HSD17B10
SCHEMBL6822414 0.74 PTGDR2 (0.36) MMP13
SCHEMBL6818697 0.72 MAPK1 (0.44) MMP13ALDH1A1HSD17B10ROCK2RPS6KA5
SCHEMBL6698728 0.70 PTGER4 (0.47) MMP13PTGER4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014916-A1 PYRIMIDINE FUSED BICYCLIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed