SCHEMBL6824523

SCHEMBL6824523

Cc1ccc(C(=O)c2ccc(OCc3ccccc3)c(-c3ccnc(NCC(=O)O)n3)c2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 6/20 0.47
CDK9 P50750 6/20 0.47
CCNA2 P20248 5/20 0.47
CDK2 P24941 5/20 0.47
CCNA1 P78396 5/20 0.47
MRGPRX4 Q96LA9 1/20 0.41
LRRK2 Q5S007 1/20 0.41
PTGER1 P34995 4/20 0.39
BRD4 O60885 1/20 0.39
SYK P43405 1/20 0.38
HDAC8 Q9BY41 2/20 0.37
DHODH Q02127 1/20 0.37
HDAC1 Q13547 2/20 0.36
SMPD1 P17405 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PTGER4 P35408 2/20 0.36
PTGER3 P43115 2/20 0.36
PTGER2 P43116 2/20 0.36
MAOB P27338 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826434 0.84 HDAC8 (0.39) CCNT1CDK9CCNA2CDK2CCNA1
SCHEMBL6823947 0.77 MRGPRX4 (0.43) MRGPRX4LRRK2PTGER1BRD4DHODH
SCHEMBL6916270 0.77 MRGPRX4 (0.41) MRGPRX4LRRK2PTGER1BRD4SYK
SCHEMBL6823543 0.76 MRGPRX4 (0.42) MRGPRX4LRRK2PTGER1BRD4DHODH
SCHEMBL6823726 0.73 MRGPRX4 (0.50) MRGPRX4LRRK2PTGER1HDAC8HDAC1
SCHEMBL6823862 0.73 HDAC8 (0.42) CCNT1CDK9CDK2HDAC8HDAC1
SCHEMBL7068093 0.72 RAF1 (0.45) CDK2MRGPRX4BRD4
SCHEMBL6820830 0.71 MRGPRX4 (0.46) MRGPRX4LRRK2PTGER1BRD4HDAC8
SCHEMBL6824812 0.70 CDK1 (0.39) CDK2BRD4
SCHEMBL6919700 0.69 MRGPRX4 (0.47) MRGPRX4LRRK2PTGER1HDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed