SCHEMBL6824813

SCHEMBL6824813

Cc1cc(-c2ccc([C@@H](O)C3(C)NC(=O)NC3=O)cc2)ccc1C#N

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 10/20 0.34
AR P10275 2/20 0.32
MGAT2 Q10469 1/20 0.31
CYP11B1 P15538 2/20 0.31
CYP11B2 P19099 2/20 0.31
EGLN2 Q96KS0 1/20 0.31
SLC2A1 P11166 1/20 0.30
PGR P06401 1/20 0.30
S1PR1 P21453 2/20 0.30
S1PR2 O95136 1/20 0.30
S1PR4 O95977 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6919077 1.00 S1PR3 (0.34) S1PR3ARMGAT2CYP11B1CYP11B2
SCHEMBL6793038 0.83 ALDH1A1 (0.41) PGR
SCHEMBL6794482 0.81 PGR (0.49) ARPGR
SCHEMBL8339982 0.78 PGR (0.41) PGR
SCHEMBL6791227 0.77 MMP2 (0.41)
SCHEMBL6789361 0.77 MMP2 (0.41)
SCHEMBL6791153 0.77 MMP2 (0.41)
SCHEMBL27584544 0.77 MCL1 (0.41) CYP11B1CYP11B2PGR
SCHEMBL6789612 0.77 PGR (0.36) ARPGR
SCHEMBL8343005 0.76 MMP3 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004024060-A2 METALLOPROTEINASE INHIBITORS AND INTERMEDIATES FOR PREPARATION THEREOF ASTRAZENECA AB (SE) 2004-03-25 WO claimed