SCHEMBL6827809

SCHEMBL6827809

Brc1cnc(NCc2ccco2)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.46
HTT P42858 3/20 0.46
LMNA P02545 2/20 0.46
MAPK1 P28482 2/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
NOD2 Q9HC29 1/20 0.46
FYN P06241 2/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 1/20 0.44
BLM P54132 1/20 0.44
POLB P06746 1/20 0.44
KCNH3 Q9ULD8 1/20 0.43
HIF1A Q16665 2/20 0.43
RAB9A P51151 2/20 0.43
DNMT1 P26358 1/20 0.42
ADRA2A P08913 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31144992 0.76 KCNH3 (0.50) SMN1; SMN2HTTLMNAMAPK1TSHR
SCHEMBL13115771 0.75 ADRA2A (0.55) SMN1; SMN2HTTLMNAMAPK1TSHR
SCHEMBL22191398 0.73 ALDH1A1 (0.57) SMN1; SMN2LMNAALDH1A1HPGDMEN1
SCHEMBL10966604 0.72 ALDH1A1 (0.62) SMN1; SMN2HTTLMNAMAPK1ALDH1A1
SCHEMBL22191568 0.70 KCNH3 (0.51) SMN1; SMN2HTTLMNAMAPK1TSHR
SCHEMBL23362392 0.70 HTT (0.48) SMN1; SMN2HTTLMNAMAPK1TSHR
SCHEMBL16381665 0.70 STIM1 (0.43) SMN1; SMN2LMNAALDH1A1HPGDMEN1
SCHEMBL5944684 0.70 POLB (0.42) SMN1; SMN2HTTLMNAMAPK1TSHR
SCHEMBL308835 0.69 TPH1 (0.52) SMN1; SMN2ALDH1A1HPGDMEN1KMT2A
SCHEMBL20119731 0.68 SMN1; SMN2 (0.46) SMN1; SMN2HTTLMNAMAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085409-A2 COMPOUNDS AND LIBRARIES OF PYRIDINES, PYRAZINES, IMIDAZO[1,2-A]PYRAZINES AND 1H-IMIDAZO[4,5-B]PYRAZIN-2-ONES AND FIRST AND SECOND MEDICAL USES THEREOF BIOFOCUS DISCOVERY LTD (GB) 2004-10-07 WO disclosed