SCHEMBL6828830

SCHEMBL6828830

CC(C)c1cc(=O)[nH]nc1-c1sc(NC(=O)COc2ccccc2)nc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.48
ADORA3 P0DMS8 4/20 0.48
RAB9A P51151 5/20 0.46
ALDH1A1 P00352 4/20 0.46
MAPT P10636 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
NPC1 O15118 3/20 0.46
TSHR P16473 2/20 0.46
HSD17B10 Q99714 2/20 0.45
MAPK1 P28482 1/20 0.45
ADORA1 P30542 6/20 0.45
TP53 P04637 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HPGD P15428 1/20 0.44
XIAP P98170 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825783 0.88 ADORA1 (0.56) ADORA2AADORA3ALDH1A1MAPTTSHR
SCHEMBL6830910 0.86 ALDH1A1 (0.46) ADORA2AADORA3ALDH1A1MAPTKDM4E
SCHEMBL6828505 0.85 ADORA2A (0.54) ADORA2AADORA3ALDH1A1MAPTADORA1
SCHEMBL6828357 0.83 ADORA2A (0.51) ADORA2AADORA3RAB9AMAPTNPC1
SCHEMBL6830218 0.83 ALDH1A1 (0.43) ADORA2AALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL6828670 0.83 XIAP (0.44) ADORA2AADORA3ALDH1A1MAPTSMN1; SMN2
SCHEMBL6826020 0.83 NPC1 (0.48) ADORA2AADORA3RAB9AALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL6828860 0.82 ALDH1A1 (0.47) ADORA2ARAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL6830646 0.82 ADORA2A (0.53) ADORA2ARAB9AALDH1A1MAPTKDM4E
SCHEMBL6828729 0.82 ADORA1 (0.57) ADORA2AADORA3RAB9AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed