SCHEMBL6828670

SCHEMBL6828670

CC(C)c1cc(=O)[nH]nc1-c1sc(NC(=O)OC(C)(C)C)nc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 5/20 0.44
ALDH1A1 P00352 4/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALOX5 P09917 1/20 0.42
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
LCK P06239 1/20 0.41
JUN P05412 1/20 0.40
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA2A P29274 4/20 0.38
ADORA1 P30542 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825783 0.83 ADORA1 (0.56) XIAPALDH1A1HSD17B10ALOX5MAPT
SCHEMBL6830646 0.83 ADORA2A (0.53) XIAPALDH1A1MAPTMEN1KMT2A
SCHEMBL6828830 0.83 ADORA2A (0.48) XIAPALDH1A1HSD17B10MAPTMEN1
SCHEMBL6828357 0.82 ADORA2A (0.51) XIAPMAPTKMT2AHTTNPSR1
SCHEMBL6828483 0.81 XIAP (0.44) XIAPALDH1A1MAPTSMN1; SMN2NPSR1
SCHEMBL6830910 0.81 ALDH1A1 (0.46) XIAPALDH1A1HSD17B10MAPTKMT2A
SCHEMBL6830337 0.81 ADORA2A (0.50) XIAPALDH1A1KMT2ALMNASMN1; SMN2
SCHEMBL6826020 0.81 NPC1 (0.48) XIAPALDH1A1KMT2ASMN1; SMN2NPSR1
SCHEMBL6828729 0.81 ADORA1 (0.57) ALDH1A1CYP2C9CYP2C19MAPTMEN1
SCHEMBL6828997 0.81 ADORA3 (0.49) XIAPALDH1A1HSD17B10MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed