SCHEMBL6829459

SCHEMBL6829459

O=C(N[C@H]1CCCC[C@H]1C(=O)O)c1ccc2ccncc2c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.54
LCK P06239 1/20 0.51
CSF1R P07333 1/20 0.51
KDR P35968 1/20 0.51
MAPK14 Q16539 1/20 0.51
AKT1 P31749 3/20 0.44
CDK2 P24941 1/20 0.43
NAMPT P43490 1/20 0.43
TAS1R3 Q7RTX0 5/20 0.43
TAS1R1 Q7RTX1 4/20 0.43
SSTR3 P32745 1/20 0.43
DRD4 P21917 1/20 0.41
TYMS P04818 1/20 0.41
TAS1R2 Q8TE23 4/20 0.41
CYP46A1 Q9Y6A2 1/20 0.41
GSK3B P49841 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5258271 1.00 SMYD3 (0.54) SMYD3LCKCSF1RKDRMAPK14
SCHEMBL5260931 0.81 AKT1 (0.44) SMYD3LCKCSF1RKDRMAPK14
SCHEMBL5258190 0.80 L3MBTL1 (0.51) NAMPTTAS1R3TAS1R1TYMSTAS1R2
SCHEMBL6832675 0.80 L3MBTL1 (0.51) NAMPTTAS1R3TAS1R1TYMSTAS1R2
SCHEMBL5404931 0.77 ROCK2 (0.54) MAPK14AKT1TYMS
SCHEMBL6829588 0.77 HTR3A (0.62) MAPK14TAS1R3TAS1R1TAS1R2
SCHEMBL5258295 0.77 HTR3A (0.62) MAPK14TAS1R3TAS1R1TAS1R2
SCHEMBL6832868 0.75 CHRNA7 (0.60) SMYD3MAPK14TAS1R3TAS1R1TYMS
SCHEMBL5254736 0.75 CHRNA7 (0.60) SMYD3MAPK14TAS1R3TAS1R1TYMS
SCHEMBL28148124 0.75 SMYD3 (0.87) SMYD3LCKCSF1RKDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6747053-B2 Heteroaryl nitriles ROCHE PALO ALTO LLC 2004-06-08 US disclosed