SCHEMBL6829470

SCHEMBL6829470

COc1c(C2CCN(C(=O)C(F)(F)F)CC2)cccc1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 10/20 0.44
MAPT P10636 3/20 0.42
MAPK1 P28482 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
SLC9A1 P19634 1/20 0.37
CYP2C19 P33261 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6829429 0.94 RBP4 (0.41) RBP4MAPTMAPK1TDP1ALDH1A1
SCHEMBL8305045 0.81 RBP4 (0.50) RBP4MEN1KMT2ACYP3A4CYP2C9
SCHEMBL28092503 0.80 TDP1 (0.46) MAPTMAPK1TDP1ALDH1A1MEN1
SCHEMBL6786475 0.76 MEN1 (0.66) RBP4MAPTALDH1A1MEN1KMT2A
SCHEMBL6791221 0.76 MAPK1 (0.47) RBP4MAPTMAPK1TDP1ALDH1A1
SCHEMBL2205192 0.74 HTR2C (0.50) MAPTMAPK1TDP1ALDH1A1
Nitric Acid SCHEMBL6720251 0.74 MAPK1 (0.46) RBP4MAPTMAPK1TDP1ALDH1A1
SCHEMBL6827413 0.74 MAPT (0.42) MAPTMAPK1TDP1ALDH1A1KMT2A
SCHEMBL9671327 0.72 HPGDS (0.44) RBP4MAPTALDH1A1MEN1KMT2A
SCHEMBL6827610 0.71 MEN1 (0.59) RBP4MAPTALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004010943-A2 SUBSTITUTED BENZANILIDES AS MODULATORS OF THE CCR5 RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2004-02-05 WO disclosed
EP-0898569-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GmbH (DE) 1999-03-03 EP disclosed
WO-1997040038-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GMBH (DE) 1997-10-30 WO disclosed