SCHEMBL6831408

SCHEMBL6831408

CC(C)[C@H](NC(=O)CCc1ccccc1)C(=O)[C@@H](C(=O)COc1c(F)c(F)cc(F)c1F)C(N)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 19/20 0.50
CASP6 P55212 19/20 0.50
CASP8 Q14790 19/20 0.50
CASP7 P55210 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419147 0.89 CASP3 (0.45) CASP3CASP6CASP8CASP7
SCHEMBL6831425 0.80 CTSV (0.45) CASP3CASP6CASP8CASP7
SCHEMBL7201965 0.79 CASP3 (0.77) CASP3CASP6CASP8CASP7
SCHEMBL7200874 0.70 CASP3 (0.40) CASP3CASP6CASP8CASP7
SCHEMBL5711363 0.70 ALDH1A1 (0.56)
SCHEMBL6446379 0.70 ALDH1A1 (0.56)
SCHEMBL7404706 0.66 CASP3 (0.57) CASP3CASP6CASP8CASP7
SCHEMBL12716161 0.66 CASP3 (0.55) CASP3CASP6CASP8CASP7
SCHEMBL25985226 0.66 KDM4E (0.52) CASP3CASP6CASP8CASP7
SCHEMBL12745894 0.66 CASP3 (0.54) CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480999-A2 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals (US) 2004-12-01 EP disclosed
WO-2003072528-A2 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2003-09-04 WO disclosed