SCHEMBL6839255

SCHEMBL6839255

CN(C#N)C(=O)[C@@H]1CCCC[C@@H]1NC(=O)c1cc2cccc(Cl)c2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.44
PYGM P11217 1/20 0.44
SMYD3 Q9H7B4 2/20 0.40
HRH4 Q9H3N8 1/20 0.40
TAS1R3 Q7RTX0 4/20 0.39
TAS1R1 Q7RTX1 4/20 0.39
TAS1R2 Q8TE23 3/20 0.39
NSD2 O96028 1/20 0.38
SETD2 Q9BYW2 1/20 0.38
PLA2G7 Q13093 4/20 0.37
KCNH2 Q12809 2/20 0.35
GHSR Q92847 2/20 0.35
MAP3K5 Q99683 1/20 0.35
OPRM1 P35372 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6839002 0.89 SMYD3 (0.40) PYGLPYGMSMYD3HRH4NSD2
SCHEMBL6838410 0.88 SMYD3 (0.40) PYGLPYGMSMYD3HRH4TAS1R3
SCHEMBL6753481 0.82 F10 (0.51) PYGLPYGMSMYD3
SCHEMBL6840639 0.82 F10 (0.51) PYGLPYGMSMYD3
SCHEMBL6382289 0.82 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2
SCHEMBL6382292 0.82 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2
SCHEMBL6839037 0.80 SMYD3 (0.34) SMYD3NSD2SETD2PLA2G7GHSR
SCHEMBL6838480 0.80 TBXAS1 (0.35) SMYD3NSD2SETD2GHSR
SCHEMBL6386703 0.79 TAS1R3 (0.56) TAS1R3TAS1R1TAS1R2KCNH2
SCHEMBL6386698 0.79 TAS1R3 (0.56) TAS1R3TAS1R1TAS1R2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759428-B2 SUCH AS N-((1,2)-2-(((CYANO(CYCLOPROPYL)METHYL)AMINO)CARBONYL) CYCLOHEXYL)-1H-INDOLE-2-CARBOXAMIDE; CATHEPSIN K INHIBITORS ROCHE PALO ALTO LLC 2004-07-06 US disclosed