SCHEMBL6840639

SCHEMBL6840639

CN(C#N)C(=O)[C@@H]1CCCC[C@@H]1NC(=O)c1cc2ccc(Cl)cc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.51
ALOX15 P16050 6/20 0.48
PYGL P06737 7/20 0.43
PYGM P11217 1/20 0.43
F2 P00734 2/20 0.42
SMYD3 Q9H7B4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6753481 1.00 F10 (0.51) F10ALOX15PYGLPYGMF2
SCHEMBL6840928 0.89 GHSR (0.41) F10
SCHEMBL6839437 0.89 DRD4 (0.50) F10ALOX15PYGLPYGM
SCHEMBL5260262 0.83 F10 (0.59) F10ALOX15PYGLPYGMF2
SCHEMBL6839255 0.82 PYGL (0.44) PYGLPYGMSMYD3
SCHEMBL6386370 0.82 TAS1R3 (0.49) F10
SCHEMBL6386374 0.82 TAS1R3 (0.49) F10
SCHEMBL6380975 0.80 TAS1R3 (0.61)
SCHEMBL6380972 0.80 TAS1R3 (0.61)
SCHEMBL16842006 0.79 TAS1R3 (0.59) F10ALOX15PYGLPYGMF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759428-B2 SUCH AS N-((1,2)-2-(((CYANO(CYCLOPROPYL)METHYL)AMINO)CARBONYL) CYCLOHEXYL)-1H-INDOLE-2-CARBOXAMIDE; CATHEPSIN K INHIBITORS ROCHE PALO ALTO LLC 2004-07-06 US disclosed