SCHEMBL6839002

SCHEMBL6839002

CN(C#N)C(=O)[C@@H]1CCCC[C@@H]1NC(=O)c1cc2cccc(Br)c2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.40
HRH4 Q9H3N8 1/20 0.40
NSD2 O96028 3/20 0.38
SETD2 Q9BYW2 2/20 0.38
PLA2G7 Q13093 9/20 0.37
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
PYGL P06737 2/20 0.33
PYGM P11217 2/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6839255 0.89 PYGL (0.44) SMYD3HRH4NSD2SETD2PLA2G7
SCHEMBL6838410 0.88 SMYD3 (0.40) SMYD3HRH4NSD2SETD2PLA2G7
SCHEMBL6839437 0.82 DRD4 (0.50) HRH4PYGLPYGM
SCHEMBL6839037 0.80 SMYD3 (0.34) SMYD3NSD2SETD2PLA2G7
SCHEMBL6838480 0.80 TBXAS1 (0.35) SMYD3NSD2SETD2
SCHEMBL6840928 0.79 GHSR (0.41)
SCHEMBL6753481 0.78 F10 (0.51) SMYD3PYGLPYGM
SCHEMBL6840639 0.78 F10 (0.51) SMYD3PYGLPYGM
SCHEMBL6385242 0.74 TAS1R3 (0.41) CNR2
SCHEMBL6382292 0.73 TAS1R3 (0.58) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759428-B2 SUCH AS N-((1,2)-2-(((CYANO(CYCLOPROPYL)METHYL)AMINO)CARBONYL) CYCLOHEXYL)-1H-INDOLE-2-CARBOXAMIDE; CATHEPSIN K INHIBITORS ROCHE PALO ALTO LLC 2004-07-06 US disclosed