SCHEMBL6839686

SCHEMBL6839686

O=[N+]([O-])c1ccc(CO[PH](=S)S)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.56
AKR1C3 P42330 1/20 0.50
LOXL2 Q9Y4K0 1/20 0.47
TSHR P16473 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAOB P27338 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP2C19 P33261 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2058333 0.80 IDO1 (0.61) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL2058336 0.77 IDO1 (0.58) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL8062311 0.75 IDO1 (0.70) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL37463 0.75 IDO1 (0.70) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL7761382 0.75 IDO1 (0.54) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL3935764 0.73 IDO1 (0.61) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL3935769 0.73 IDO1 (0.61) IDO1AKR1C3LOXL2TSHRCA12
Butane SCHEMBL8720911 0.72 IDO1 (0.51) IDO1AKR1C3LOXL2TSHRMEN1
SCHEMBL23091915 0.72 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12
SCHEMBL21753899 0.72 IDO1 (0.66) IDO1AKR1C3LOXL2TSHRCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756496-B1 SUCH AS TRIETHYLAMMONIUM-5'-DIMETHOXYTRITYL-3'-THYMIDINE-HYDROGEN PHOSPHONONDITHIOATE FOR USE AS ANTIVIRAL AND ANTICANCER AGENTS ISIS PHARMACEUTICALS, INC. 2004-06-29 US disclosed
US-5565555-A Nucleoside hydrogen phosphonodithioate diesters and activated phosphonodithioate analogues GILEAD SCIENCES, INC. (US) 1996-10-15 US disclosed
US-5194599-A Forming linkages with nuclosides and nucleotides; viricides, anticarcinogenic agents GILEAD SCIENCES, INC. (US) 1993-03-16 US disclosed
EP-0360609-A2 Novel hydrogen phosphonodithioate compositions GILEAD SCIENCES, INC. (US) 1990-03-28 EP disclosed