SCHEMBL6844957

SCHEMBL6844957

Cc1cc(-c2cccnc2)ncn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 7/20 0.62
KMO O15229 1/20 0.59
CYP3A4 P08684 9/20 0.56
CYP1A2 P05177 7/20 0.56
CLK4 Q9HAZ1 5/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CYP2C19 P33261 6/20 0.54
HSD17B10 Q99714 5/20 0.54
CYP2D6 P10635 4/20 0.54
TSHR P16473 2/20 0.54
ALOX15 P16050 1/20 0.54
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 1/20 0.52
HPGD P15428 1/20 0.52
CYP2E1 P05181 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2B6 P20813 2/20 0.51
ALK Q9UM73 1/20 0.51
PIM1 P11309 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18905235 0.81 KMO (0.68) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL2129077 0.79 ASIC3 (0.59) KMOCYP1A2MEN1KMT2ACYP2C19
SCHEMBL30412356 0.79 ASIC3 (0.59) KMOCYP1A2MEN1KMT2ACYP2C19
SCHEMBL1444763 0.79 MIF (0.65) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL31205777 0.79 KMO (0.59) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL24151512 0.79 KMO (0.59) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL558195 0.79 ASIC3 (0.65) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL30507429 0.79 ASIC3 (0.65) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL20816293 0.78 CYP1A2 (0.62) CYP2A6KMOCYP3A4CYP1A2CLK4
SCHEMBL10220550 0.78 KMO (0.55) CYP2A6KMOCYP3A4CYP1A2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9666807-B2 Organic light emitting device SAMSUNG DISPLAY CO., LTD. (KR) 2017-05-30 US disclosed
US-9666807-B2 Organic light emitting device SAMSUNG DISPLAY CO., LTD. (KR) 2017-05-30 US disclosed
US-20160101104-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL MYERS SQUIBB CO (US) 2016-04-14 US disclosed
US-20160028017-A1 ORGANIC LIGHT EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2016-01-28 US disclosed
US-20150342935-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL MYERS SQUIBB CO (US) 2015-12-03 US disclosed
US-20150094309-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL MYERS SQUIBB CO (US) 2015-04-02 US disclosed
US-20140221377-A1 Quinuclidine Compounds as Alpha-7 Nicotinic Acetylcholine Receptor Ligands BRISTOL MYERS SQUIBB CO (US) 2014-08-07 US disclosed
WO-2011053292-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-05 WO disclosed
WO-2009131926-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-10-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221377-A1 Quinuclidine Compounds as Alpha-7 Nicotinic Acetylcholine Receptor Ligands CHRNA7, CHRNA5, CHRNA6 CYP2A6 2357/4885KMO 932/4885CYP3A4 2815/4885
US-20160101104-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS CHRNA7, CHRNA5, CHRNA6 CYP2A6 2357/4885KMO 932/4885CYP3A4 2815/4885
US-20150342935-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS CHRNA7, CHRNA5, CHRNA6 CYP2A6 2357/4885KMO 932/4885CYP3A4 2815/4885
US-20150094309-A1 QUINUCLIDINE COMPOUNDS AS ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS CHRNA7, CHRNA5, CHRNA6 CYP2A6 2357/4885KMO 932/4885CYP3A4 2815/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.