SCHEMBL6845271

SCHEMBL6845271

CNC(C)c1ccc(C(=O)Nc2ccnc([N+](=O)[O-])c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 2/20 0.44
MAPT P10636 9/20 0.42
POLB P06746 2/20 0.42
MAPK1 P28482 2/20 0.42
MITF O75030 1/20 0.42
RAB9A P51151 7/20 0.42
KMT2A Q03164 5/20 0.41
USP2 O75604 1/20 0.41
NPC1 O15118 5/20 0.41
MEN1 O00255 4/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 2/20 0.41
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6845274 0.81 ROCK2 (0.48) ROCK2ROCK1MAPTRAB9AKMT2A
SCHEMBL27500826 0.80 MEN1 (0.56) MAPTPOLBMITFRAB9AKMT2A
SCHEMBL6845275 0.80 ROCK2 (0.47) ROCK2ROCK1RAB9ANPC1ALDH1A1
SCHEMBL6845267 0.77 ROCK2 (0.71) ROCK2ROCK1MAPTPOLBMAPK1
SCHEMBL6845277 0.77 ROCK2 (0.44) ROCK2ROCK1RAB9AKMT2ANPC1
SCHEMBL16964837 0.72 POLB (0.56) MAPTPOLBMAPK1MITFRAB9A
SCHEMBL6557961 0.68 ROCK2 (0.68) ROCK2ROCK1MAPTPOLBMAPK1
SCHEMBL11621907 0.68 MAPT (0.54) MAPTPOLBMAPK1MITFKMT2A
SCHEMBL1880283 0.66 ALDH1A1 (0.50) MAPTMAPK1RAB9AKMT2ANPC1
SCHEMBL11618215 0.66 KMT2A (0.41) MAPTPOLBMAPK1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7867999-B1 Hydroxyamino- and amino-substituted pyridine analogs for treating rho kinase-mediated diseases and conditions ALCON RESEARCH, LTD. (US) 2011-01-11 US disclosed