SCHEMBL6848796

SCHEMBL6848796

COc1cc(Cl)cc(NC(=N)N(C)c2cccc([S+](C)[O-])c2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
P2RX1 P51575 1/20 0.32
PTGS2 P35354 1/20 0.32
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
POLB P06746 2/20 0.32
HTT P42858 2/20 0.31
MAPT P10636 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7745766 0.99 HTR3E (0.34) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6847040 0.83 P2RX7 (0.37) HSD17B1HSD17B2POLBHTTMAPT
Hydrochloric Acid SCHEMBL7743900 0.82 P2RX7 (0.36) HSD17B1HSD17B2POLBHTTMAPT
SCHEMBL6720863 0.73 GAA (0.41) MAPTMAPK1SMN1; SMN2
SCHEMBL6846356 0.73 GRIN2D (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL499302 0.73 GRIN2D (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL499303 0.73 GRIN2D (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL7743328 0.72 GRIN2D (0.43) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8194423 0.71 SIGMAR1 (0.43) MAPTMEN1KMT2A
SCHEMBL6847741 0.71 MAPT (0.37) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6774263-B1 N-(2-CHLORO-5-METHYLTHIOPHENYL)-N'-(3-METHYLSULFINYLPHENYL)-N' -METHYLGUANIDINE; NEURODEGENERATIVE DISORDER TREATMENT CAMBRIDGE NEUROSCIENCE, INC. 2004-08-10 US disclosed