SCHEMBL6854224

SCHEMBL6854224

Cc1ccc(-c2ccc(/C=C/CO)cc2)nn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
CYP3A4 P08684 2/20 0.39
RECQL P46063 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.34
NPC1 O15118 4/20 0.34
RAB9A P51151 4/20 0.34
LMNA P02545 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
APLNR P35414 1/20 0.33
P2RX7 Q99572 2/20 0.33
KDM4E B2RXH2 4/20 0.33
HPGD P15428 4/20 0.33
MITF O75030 1/20 0.33
KLF5 Q13887 1/20 0.33
CASP3 P42574 1/20 0.31
SENP8 Q96LD8 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6854227 1.00 ALDH1A1 (0.39) ALDH1A1CYP3A4RECQLSMN1; SMN2NPC1
SCHEMBL6852515 0.81 LMNA (0.40) ALDH1A1CYP3A4RECQLSMN1; SMN2NPC1
SCHEMBL6852522 0.81 LMNA (0.40) ALDH1A1CYP3A4RECQLSMN1; SMN2NPC1
SCHEMBL6852317 0.78 APLNR (0.36) CYP3A4SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL17051575 0.76 NPC1 (0.44) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA
SCHEMBL6851881 0.75 HDAC4 (0.43) ALDH1A1CYP3A4RECQLP2RX7
SCHEMBL6851894 0.75 HDAC4 (0.43) ALDH1A1CYP3A4RECQLP2RX7
SCHEMBL12970083 0.74 FYN (0.41) SMN1; SMN2NPC1RAB9ALMNANFKB1
SCHEMBL26018390 0.74 KDM4E (0.33) ALDH1A1SMN1; SMN2NPC1RAB9AAPLNR
SCHEMBL7029497 0.72 GPR119 (0.34) ALDH1A1SMN1; SMN2NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed