SCHEMBL6854936

SCHEMBL6854936

Cc1c(CC(=O)NC(C)C)c(-c2ccc(F)c(Cl)c2)nc2ccc(N3CCC(=O)CC3)cc12

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 12/20 0.41
ACACB O00763 2/20 0.38
ENPP2 Q13822 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
MCHR1 Q99705 1/20 0.36
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6856891 0.90 AVPR1B (0.40) AVPR1BACACBENPP2MCHR1
SCHEMBL6857500 0.88 AVPR1B (0.41) AVPR1BACACBENPP2MCHR1
SCHEMBL6856813 0.87 AVPR1B (0.40) AVPR1BACACBENPP2CASP3
SCHEMBL6855979 0.83 AVPR1B (0.39) AVPR1B
SCHEMBL6856235 0.82 AVPR1B (0.39) AVPR1B
SCHEMBL6857461 0.81 AVPR1B (0.44) AVPR1BACACB
SCHEMBL6857432 0.79 AVPR1B (0.43) AVPR1B
SCHEMBL6856705 0.79 AVPR1B (0.58) AVPR1B
SCHEMBL6856801 0.79 HRH3 (0.43) AVPR1BACACB
SCHEMBL6857472 0.77 AVPR1B (0.51) AVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed