SCHEMBL6855979

SCHEMBL6855979

Cc1c(CC(=O)NC(C)C)c(-c2ccc(F)c(Cl)c2)nc2ccc(O)cc12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 3/20 0.39
ESR1 P03372 4/20 0.38
ESR2 Q92731 4/20 0.38
CTSA P10619 3/20 0.38
DHODH Q02127 2/20 0.38
TSPO P30536 1/20 0.37
ABL1 P00519 1/20 0.36
SLC1A3 P43003 1/20 0.36
SLC1A2 P43004 1/20 0.36
SLC1A1 P43005 1/20 0.36
ICMT O60725 1/20 0.36
CNR2 P34972 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
ESRRB O95718 1/20 0.36
ESRRA P11474 1/20 0.36
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6856235 0.89 AVPR1B (0.39) AVPR1BCTSADHODHTSPOABL1
SCHEMBL6856869 0.87 AVPR1B (0.45) AVPR1BESRRBESRRA
SCHEMBL6857432 0.85 AVPR1B (0.43) AVPR1BICMT
SCHEMBL6857370 0.83 TRPV1 (0.39) AVPR1BCTSAABL1SLC1A3SLC1A2
SCHEMBL6854936 0.83 AVPR1B (0.41) AVPR1B
SCHEMBL6856891 0.81 AVPR1B (0.40) AVPR1BKDM4E
SCHEMBL6856705 0.80 AVPR1B (0.58) AVPR1BESR1
SCHEMBL6856801 0.80 HRH3 (0.43) AVPR1B
SCHEMBL6857500 0.80 AVPR1B (0.41) AVPR1B
SCHEMBL6856813 0.79 AVPR1B (0.40) AVPR1BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed