SCHEMBL6856940

SCHEMBL6856940

Bc1ccc2nc(-c3cccc(Cl)c3)c(CC(=O)O)cc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.41
RXRB P28702 2/20 0.41
RXRG P48443 2/20 0.41
KDM4E B2RXH2 3/20 0.40
FFAR1 O14842 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NR4A2 P43354 1/20 0.39
AVPR1A P37288 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PDE4B Q07343 2/20 0.38
PDE4D Q08499 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
TYMP P19971 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857026 0.84 AVPR1B (0.48)
SCHEMBL6856769 0.84 KMO (0.39) KDM4EMEN1KMT2AALDH1A1PTGDR2
SCHEMBL6856938 0.84 PTGDR2 (0.44) RXRARXRBKDM4ECSNK2A2CSNK2B
SCHEMBL10102664 0.82 KDM4E (0.50) KDM4EMEN1KMT2AALDH1A1CYP2C19
SCHEMBL6857165 0.79 KDM4E (0.51) RXRARXRBRXRGKDM4EMEN1
SCHEMBL10509302 0.72 KDM4E (0.65) KDM4EMEN1KMT2ANR4A2ALDH1A1
SCHEMBL3384876 0.72 KDM4E (0.53) KDM4EMEN1KMT2AALDH1A1LMNA
SCHEMBL6857065 0.69 AVPR1B (0.45) AVPR1A
SCHEMBL6857380 0.69 TRPV1 (0.38) KDM4E
SCHEMBL6857381 0.69 MDM2 (0.40) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed