SCHEMBL6856769

SCHEMBL6856769

Bc1ccc2nc(-c3ccc(F)c(Cl)c3)c(CC(=O)O)cc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.39
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
DGAT1 O75907 1/20 0.36
RPA1 P27694 1/20 0.36
ICMT O60725 1/20 0.35
PTGDR2 Q9Y5Y4 3/20 0.35
TBXA2R P21731 1/20 0.35
PTGDR Q13258 1/20 0.35
MDM2 Q00987 1/20 0.35
CASP3 P42574 1/20 0.35
TSPO P30536 1/20 0.35
CTSA P10619 1/20 0.35
HPSE Q9Y251 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
DHODH Q02127 1/20 0.34
FABP4 P15090 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6856809 0.84 MTNR1A (0.36) KMOICMTCASP3TSPOCTSA
SCHEMBL6857380 0.84 TRPV1 (0.38) ICMTCTSAKDM4E
SCHEMBL6857381 0.84 MDM2 (0.40) ICMTMDM2
SCHEMBL6856940 0.84 RXRA (0.41) KMOPTGDR2TBXA2RPTGDRKDM4E
SCHEMBL6856237 0.82 KMO (0.42) KMOADORA2AADORA1DGAT1RPA1
SCHEMBL6856907 0.81 LMNA (0.43) KMOPTGDR2MDM2CASP3TSPO
SCHEMBL6856938 0.75 PTGDR2 (0.44) ADORA2APTGDR2KDM4EALDH1A1
SCHEMBL6856613 0.75 HRH3 (0.48) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL10102664 0.73 KDM4E (0.50) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL6856772 0.72 MTNR1A (0.36) KMOCASP3TSPOKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed