SCHEMBL6857475

SCHEMBL6857475

COc1cccc(-c2nc3ccc(OCCCN4CCOCC4)cc3cc2CC(=O)NC(C)C)n1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 14/20 0.54
HRH3 Q9Y5N1 1/20 0.47
MIF P14174 1/20 0.46
EPHX2 P34913 1/20 0.44
ATM Q13315 1/20 0.44
ROCK1 Q13464 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857173 0.92 AVPR1B (0.45) AVPR1BHRH3
SCHEMBL6856961 0.85 SMN1; SMN2 (0.39) AVPR1B
SCHEMBL6855518 0.84 AVPR1B (0.66) AVPR1BHRH3
SCHEMBL16423582 0.80 AVPR1B (0.61) AVPR1BHRH3
SCHEMBL6856187 0.80 AVPR1B (0.65) AVPR1BHRH3
SCHEMBL6856988 0.80 AVPR1B (0.53) AVPR1BHRH3MIFATM
SCHEMBL6856966 0.78 PTGES (0.39) AVPR1B
SCHEMBL6857205 0.77 AVPR1B (0.65) AVPR1B
SCHEMBL6857155 0.76 AVPR1B (0.56) AVPR1B
SCHEMBL16442055 0.75 AVPR1B (0.55) AVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed