SCHEMBL6858091

SCHEMBL6858091

Cc1cccc(CN2CCN(c3ccccc3)CC2)c1

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.76
KDM4E B2RXH2 3/20 0.76
MAPT P10636 1/20 0.76
DRD4 P21917 2/20 0.70
KCNH2 Q12809 1/20 0.62
DRD2 P14416 2/20 0.60
DRD3 P35462 1/20 0.60
LMNA P02545 2/20 0.59
HPGD P15428 1/20 0.59
ALOX15 P16050 1/20 0.59
HTR7 P34969 1/20 0.59
FAAH O00519 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15938014 0.87 HTR7 (0.67) ALDH1A1KDM4EMAPTDRD4KCNH2
SCHEMBL13637639 0.85 ALDH1A1 (0.65) ALDH1A1KDM4EMAPTDRD4KCNH2
SCHEMBL7995650 0.85 HTR1A (0.71) ALDH1A1KDM4EMAPTKCNH2DRD2
SCHEMBL15359164 0.84 DRD4 (0.70) ALDH1A1KDM4EMAPTDRD4DRD2
SCHEMBL6031812 0.83 DRD4 (1.00) ALDH1A1KDM4EDRD4DRD2DRD3
SCHEMBL7498974 0.83 DRD4 (0.72) DRD4DRD2DRD3HTR7FAAH
SCHEMBL15937926 0.82 MAPT (0.61) ALDH1A1KDM4EMAPTDRD4DRD2
SCHEMBL6865778 0.82 KDM4E (0.67) ALDH1A1KDM4EMAPTLMNAALOX15
SCHEMBL7604485 0.82 DRD4 (0.77) ALDH1A1KDM4EMAPTDRD4DRD2
SCHEMBL12385909 0.82 DRD4 (0.77) ALDH1A1KDM4EMAPTDRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed
WO-1998008091-A1 NORMALIZATION OF COMBINATORIAL REACTIONS ISIS PHARMACEUTICALS, INC. (US) 1998-02-26 WO disclosed
WO-1998005332-A1 NOVEL HETEROCYCLE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 1998-02-12 WO disclosed