SCHEMBL6861498

SCHEMBL6861498

CN(C)C(=O)c1cccc(Cn2nc(C(F)(F)F)c3c2OCCC3)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 6/20 0.44
CYP2D6 P10635 2/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.43
MAPT P10636 6/20 0.41
CYP2C9 P11712 3/20 0.41
POLQ O75417 1/20 0.40
CYP2C19 P33261 2/20 0.40
DRD2 P14416 1/20 0.38
FAAH O00519 1/20 0.37
MGLL Q99685 1/20 0.37
TP53 P04637 2/20 0.36
LMNA P02545 1/20 0.36
ALDH1A1 P00352 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861342 0.88 GRIA2 (0.54) GRIA2CYP2D6CYP1A2POLBMAPT
SCHEMBL6861147 0.87 ABHD6 (0.48) POLBMAPTTP53LMNA
SCHEMBL6861702 0.87 MAPT (0.43) GRIA2CYP1A2POLBMAPTCYP2C19
SCHEMBL6864318 0.85 KDM4E (0.44) GRIA2POLBMAPTLMNAALDH1A1
SCHEMBL1007660 0.84 GRIA2 (0.57) GRIA2CYP2D6CYP1A2POLBMAPT
SCHEMBL6860475 0.78 LMNA (0.44) GRIA2CYP1A2POLBMAPTCYP2C9
SCHEMBL6860844 0.75 CYP2C19 (0.43) GRIA2CYP2D6CYP1A2POLBMAPT
SCHEMBL1006841 0.75 POLB (0.51) GRIA2CYP2D6CYP1A2POLBMAPT
SCHEMBL12998713 0.75 GRIA2 (0.69) GRIA2CYP2D6CYP1A2MAPTCYP2C9
SCHEMBL1006269 0.74 GRIA2 (0.55) GRIA2CYP2D6CYP1A2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011036889-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2011-03-31 WO disclosed