SCHEMBL6861342

SCHEMBL6861342

CN(C)C(=O)c1ccc(Cn2nc(C(F)(F)F)c3c2OCCC3)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 7/20 0.54
CYP1A2 P05177 4/20 0.54
CYP2D6 P10635 3/20 0.54
CYP2C9 P11712 4/20 0.45
CYP2C19 P33261 4/20 0.44
POLQ O75417 1/20 0.42
MAPT P10636 5/20 0.41
POLB P06746 1/20 0.41
TP53 P04637 2/20 0.39
CYP3A4 P08684 1/20 0.39
LMNA P02545 3/20 0.39
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861498 0.88 GRIA2 (0.44) GRIA2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6860475 0.87 LMNA (0.44) GRIA2CYP1A2CYP2C9CYP2C19POLQ
SCHEMBL6860844 0.84 CYP2C19 (0.43) GRIA2CYP1A2CYP2D6CYP2C19MAPT
SCHEMBL12998713 0.82 GRIA2 (0.69) GRIA2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6862770 0.82 SMN1; SMN2 (0.39) GRIA2CYP1A2CYP2D6CYP2C19MAPT
SCHEMBL6861147 0.77 ABHD6 (0.48) MAPTPOLBTP53LMNATSHR
SCHEMBL6861702 0.77 MAPT (0.43) GRIA2CYP1A2CYP2C19MAPTPOLB
SCHEMBL6864318 0.75 KDM4E (0.44) GRIA2MAPTPOLBLMNANPSR1
SCHEMBL12997891 0.74 GRIA2 (0.74) GRIA2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL15491619 0.74 LMNA (0.48) GRIA2CYP1A2CYP2C19POLQMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011036889-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2011-03-31 WO disclosed