SCHEMBL6860844

SCHEMBL6860844

CC(C)NC(=O)c1ccc(Cn2nc(C(F)(F)F)c3c2OCCC3)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 1/20 0.43
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
MAPT P10636 6/20 0.42
POLB P06746 2/20 0.41
PTGER4 P35408 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
TP53 P04637 2/20 0.40
CYP3A4 P08684 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
GRIA2 P42262 2/20 0.40
MLYCD O95822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6864318 0.89 KDM4E (0.44) MAPTPOLBPTGER4SMN1; SMN2MEN1
SCHEMBL6860475 0.86 LMNA (0.44) CYP2C19CYP1A2MAPTPOLBSMN1; SMN2
SCHEMBL6861342 0.84 GRIA2 (0.54) CYP2C19CYP1A2CYP2D6MAPTPOLB
SCHEMBL6862770 0.84 SMN1; SMN2 (0.39) CYP2C19CYP1A2CYP2D6HDAC4HDAC1
SCHEMBL6861147 0.79 ABHD6 (0.48) MAPTPOLBSMN1; SMN2TP53MEN1
SCHEMBL6861702 0.79 MAPT (0.43) CYP2C19CYP1A2MAPTPOLBSMN1; SMN2
SCHEMBL12998073 0.75 GRIA2 (0.54) CYP2C19CYP1A2CYP2D6HDAC4HDAC6
SCHEMBL6861498 0.75 GRIA2 (0.44) CYP2C19CYP1A2CYP2D6MAPTPOLB
SCHEMBL1009106 0.74 GRIA2 (0.54) CYP2C19CYP1A2MAPTPOLBSMN1; SMN2
SCHEMBL15491619 0.73 LMNA (0.48) CYP2C19CYP1A2MAPTSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011036889-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2011-03-31 WO disclosed