SCHEMBL6863248

SCHEMBL6863248

Cc1cc(NC(=O)NC2CCN(C(=O)[C@H]3CCCCN3)CC2)cc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 3/20 0.51
EPHX2 P34913 13/20 0.50
PAK3 O75914 1/20 0.45
PAK1 Q13153 1/20 0.45
PAK2 Q13177 1/20 0.45
UBE2M P61081 3/20 0.45
DCUN1D1 Q96GG9 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12004739 0.93 CXCR3 (0.55) CXCR3EPHX2PAK3PAK1PAK2
SCHEMBL6863633 0.93 CXCR3 (0.55) CXCR3EPHX2PAK3PAK1PAK2
SCHEMBL6864238 0.93 CXCR3 (0.55) CXCR3EPHX2PAK3PAK1PAK2
SCHEMBL6863225 0.90 EPHX2 (0.47) EPHX2MEN1KMT2A
SCHEMBL6863176 0.83 S1PR2 (0.40) CXCR3
SCHEMBL6863181 0.81 S1PR2 (0.41)
SCHEMBL25993053 0.80 EPHX2 (0.67) CXCR3EPHX2
SCHEMBL12005295 0.79 CXCR3 (0.46) CXCR3EPHX2PAK3PAK1PAK2
SCHEMBL12005297 0.79 CXCR3 (0.46) CXCR3EPHX2PAK3PAK1PAK2
SCHEMBL12005445 0.79 CXCR3 (0.46) CXCR3EPHX2PAK3PAK1PAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011032291-A1 SELECTIVE CALCIUM CHANNEL MODULATORS ZALICUS PHARMACEUTICALS LTD . (CA) 2011-03-24 WO disclosed