SCHEMBL6863176

SCHEMBL6863176

Cc1cc(NC(=O)NCC2(O)CCN(C(=O)[C@@H]3CCCCN3)CC2)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 7/20 0.40
CCR3 P51677 2/20 0.36
CXCR3 P49682 3/20 0.36
MAPT P10636 1/20 0.35
CYP2D6 P10635 1/20 0.35
KDR P35968 1/20 0.35
TACR1 P25103 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863132 0.94 S1PR2 (0.40) S1PR2CCR3CXCR3MAPTCYP2D6
SCHEMBL6863244 0.94 S1PR2 (0.40) S1PR2CCR3CXCR3MAPTCYP2D6
SCHEMBL6863253 0.91 CCR3 (0.38) CCR3MAPT
SCHEMBL6863181 0.90 S1PR2 (0.41) S1PR2TACR1
SCHEMBL6863172 0.89 S1PR2 (0.37) S1PR2CCR3CXCR3CYP2D6KDR
SCHEMBL6863248 0.83 CXCR3 (0.51) CXCR3
SCHEMBL6863044 0.83 S1PR2 (0.41) S1PR2
SCHEMBL12005722 0.83 S1PR2 (0.41) S1PR2
SCHEMBL6863109 0.83 S1PR2 (0.41) S1PR2
SCHEMBL12005445 0.79 CXCR3 (0.46) CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011032291-A1 SELECTIVE CALCIUM CHANNEL MODULATORS ZALICUS PHARMACEUTICALS LTD . (CA) 2011-03-24 WO disclosed