SCHEMBL6863181

SCHEMBL6863181

Cc1cc(NC(=O)CC2(O)CCN(C(=O)[C@H]3CCCCN3)CC2)cc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 7/20 0.41
P2RX7 Q99572 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TACR1 P25103 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
WNT3 P56703 2/20 0.34
SFRP1 Q8N474 2/20 0.34
PARP1 P09874 2/20 0.34
CCR4 P51679 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863109 0.94 S1PR2 (0.41) S1PR2P2RX7ALDH1A1WNT3SFRP1
SCHEMBL6863044 0.94 S1PR2 (0.41) S1PR2P2RX7ALDH1A1WNT3SFRP1
SCHEMBL12005722 0.94 S1PR2 (0.41) S1PR2P2RX7ALDH1A1WNT3SFRP1
SCHEMBL6863176 0.90 S1PR2 (0.40) S1PR2TACR1
SCHEMBL12015159 0.85 ALDH1A1 (0.40) S1PR2P2RX7ALDH1A1WNT3SFRP1
SCHEMBL12015288 0.85 ALDH1A1 (0.40) S1PR2P2RX7ALDH1A1WNT3SFRP1
SCHEMBL6863132 0.83 S1PR2 (0.40) S1PR2P2RX7
SCHEMBL6863244 0.83 S1PR2 (0.40) S1PR2P2RX7
SCHEMBL6863248 0.81 CXCR3 (0.51)
SCHEMBL6863253 0.79 CCR3 (0.38) CCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011032291-A1 SELECTIVE CALCIUM CHANNEL MODULATORS ZALICUS PHARMACEUTICALS LTD . (CA) 2011-03-24 WO disclosed