SCHEMBL6863423

SCHEMBL6863423

CCCCN(Cc1ccccc1)C(=O)c1cc(N)n2nc(-c3ccc(OC)s3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.43
HDAC1 Q13547 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
LPAR1 Q92633 6/20 0.39
LPAR2 Q9HBW0 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
LIMK1 P53667 1/20 0.39
LIMK2 P53671 1/20 0.39
LPAR5 Q9H1C0 1/20 0.39
LPAR3 Q9UBY5 1/20 0.38
PKM P14618 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
CYP3A4 P08684 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870566 0.92 ADORA2A (0.45) ADORA2ACYP2D6CYP3A4
SCHEMBL6863393 0.92 ADORA2A (0.50) ADORA2ALPAR1LPAR2LPAR5LPAR3
SCHEMBL6863124 0.92 ADORA2A (0.49) ADORA2ALPAR1LPAR5CYP3A4
SCHEMBL6867221 0.91 ADORA2A (0.46) ADORA2ALPAR1LPAR2LIMK2CYP3A4
SCHEMBL6871694 0.85 ADORA2A (0.44) ADORA2APARP1
SCHEMBL6871816 0.84 ADORA2A (0.57) ADORA2A
SCHEMBL6870537 0.83 ADORA2A (0.62) ADORA2ALTB4R2
SCHEMBL6873020 0.80 ADORA2A (0.53) ADORA2AHDAC1HDAC6CYP2D6CYP2C9
SCHEMBL6863381 0.80 ADORA2A (0.46) ADORA2ALPAR1LPAR5
SCHEMBL6867557 0.80 ADORA2A (0.46) ADORA2AHDAC1HDAC6CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed