SCHEMBL6863124

SCHEMBL6863124

CCN(Cc1ccccc1)C(=O)c1cc(N)n2nc(-c3ccc(OC)s3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.49
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LPAR1 Q92633 1/20 0.38
LPAR5 Q9H1C0 1/20 0.38
PPARG P37231 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
F2 P00734 1/20 0.36
CYP3A4 P08684 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870566 0.95 ADORA2A (0.45) ADORA2AMEN1KMT2AKDM4EALDH1A1
SCHEMBL6867221 0.92 ADORA2A (0.46) ADORA2AMEN1KMT2ALPAR1KDM4E
SCHEMBL6863423 0.92 ADORA2A (0.43) ADORA2ALPAR1LPAR5CYP3A4
SCHEMBL6863393 0.91 ADORA2A (0.50) ADORA2AMEN1KMT2ALPAR1LPAR5
SCHEMBL6871816 0.91 ADORA2A (0.57) ADORA2ALMNAHPGD
SCHEMBL6863381 0.88 ADORA2A (0.46) ADORA2ALPAR1LPAR5KDM4EALDH1A1
SCHEMBL6871694 0.88 ADORA2A (0.44) ADORA2AMEN1KMT2APPARGLMNA
SCHEMBL6870537 0.84 ADORA2A (0.62) ADORA2A
SCHEMBL6871983 0.83 ADORA2A (0.46) ADORA2ALMNAGAA
SCHEMBL6863086 0.81 PLAU (0.44) ADORA2AKDM4EALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed