SCHEMBL6870566

SCHEMBL6870566

COc1ccc(-c2nc3cc(C(=O)N(Cc4ccccc4)Cc4ccccc4)cc(N)n3n2)s1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.45
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TSHR P16473 2/20 0.39
CYP3A4 P08684 2/20 0.38
CFTR P13569 1/20 0.37
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 1/20 0.36
MEN1 O00255 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HSD17B2 P37059 2/20 0.36
HSD17B1 P14061 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863124 0.95 ADORA2A (0.49) ADORA2AKDM4ETDP1ALDH1A1LMNA
SCHEMBL6863393 0.94 ADORA2A (0.50) ADORA2ACYP3A4KMT2AMEN1
SCHEMBL6867221 0.93 ADORA2A (0.46) ADORA2AKDM4ETDP1ALDH1A1LMNA
SCHEMBL6863423 0.92 ADORA2A (0.43) ADORA2ACYP3A4CYP2D6
SCHEMBL6871694 0.90 ADORA2A (0.44) ADORA2ALMNAGAAMAPTTSHR
SCHEMBL6871816 0.88 ADORA2A (0.57) ADORA2ALMNAHPGDTSHR
SCHEMBL6870537 0.86 ADORA2A (0.62) ADORA2AHSD17B2HSD17B1
SCHEMBL6863381 0.84 ADORA2A (0.46) ADORA2AKDM4EALDH1A1LMNAMAPT
SCHEMBL6863086 0.83 PLAU (0.44) ADORA2AKDM4EALDH1A1LMNAHPGD
SCHEMBL6863519 0.83 ADORA2A (0.44) ADORA2AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed