SCHEMBL6867221

SCHEMBL6867221

COc1ccc(-c2nc3cc(C(=O)N(CCN(C)C)Cc4ccccc4)cc(N)n3n2)s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.46
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.38
LIMK2 P53671 1/20 0.38
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
POLB P06746 1/20 0.37
LPAR1 Q92633 2/20 0.36
LPAR2 Q9HBW0 1/20 0.36
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870566 0.93 ADORA2A (0.45) ADORA2AMEN1KMT2ACYP3A4KDM4E
SCHEMBL6863393 0.92 ADORA2A (0.50) ADORA2AMEN1KMT2ACYP3A4LPAR1
SCHEMBL6863124 0.92 ADORA2A (0.49) ADORA2AMEN1KMT2ACYP3A4LPAR1
SCHEMBL6863423 0.91 ADORA2A (0.43) ADORA2ACYP3A4LIMK2LPAR1LPAR2
SCHEMBL6870537 0.85 ADORA2A (0.62) ADORA2AHSD17B2HSD17B1ROCK2ROCK1
SCHEMBL6871694 0.85 ADORA2A (0.44) ADORA2AMEN1KMT2ATP53LMNA
SCHEMBL6871816 0.85 ADORA2A (0.57) ADORA2ALMNAHPGD
SCHEMBL6863381 0.81 ADORA2A (0.46) ADORA2ATP53LPAR1KDM4EALDH1A1
SCHEMBL6863086 0.79 PLAU (0.44) ADORA2ATP53KDM4EALDH1A1LMNA
SCHEMBL6863519 0.79 ADORA2A (0.44) ADORA2AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed