SCHEMBL6863381

SCHEMBL6863381

CCN(Cc1ccccc1F)C(=O)c1cc(N)n2nc(-c3ccc(OC)s3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.46
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
TSPO P30536 1/20 0.35
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
LPAR1 Q92633 2/20 0.33
HSD17B10 Q99714 3/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MCTS1 Q9ULC4 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
LPAR5 Q9H1C0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863124 0.88 ADORA2A (0.49) ADORA2AMAPTLPAR1KDM4EALDH1A1
SCHEMBL6871816 0.88 ADORA2A (0.57) ADORA2AHPGDLMNATSHR
SCHEMBL6870566 0.84 ADORA2A (0.45) ADORA2AMAPTKDM4EALDH1A1HPGD
SCHEMBL6867221 0.81 ADORA2A (0.46) ADORA2AMAPTTP53ROCK2ROCK1
SCHEMBL6863423 0.80 ADORA2A (0.43) ADORA2ALPAR1LPAR5
SCHEMBL6863393 0.80 ADORA2A (0.50) ADORA2ALPAR1LPAR5
SCHEMBL6871983 0.80 ADORA2A (0.46) ADORA2ALMNATSHR
SCHEMBL6867466 0.80 ADORA2A (0.49) ADORA2ATSPOROCK2ROCK1HSD17B10
SCHEMBL6869841 0.79 ADORA2A (0.48) ADORA2AMAPTTSPOHSD17B10KDM4E
SCHEMBL6871694 0.78 ADORA2A (0.44) ADORA2AMAPTSMN1; SMN2TP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed