SCHEMBL6863684

SCHEMBL6863684

COc1ccc(NS(C)(=O)=O)cc1C#N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
PGR P06401 2/20 0.56
NR3C1 P04150 1/20 0.53
NR3C2 P08235 1/20 0.53
AR P10275 1/20 0.53
SLC22A12 Q96S37 1/20 0.52
KDM4E B2RXH2 2/20 0.50
USP2 O75604 1/20 0.50
PLA2G7 Q13093 3/20 0.46
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KDM1A O60341 1/20 0.45
CYP17A1 P05093 4/20 0.45
HSP90AA1 P07900 2/20 0.45
HSP90AB1 P08238 2/20 0.45
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13065706 0.83 SLC22A12 (0.43) ALDH1A1PGRNR3C1NR3C2AR
SCHEMBL6857824 0.80 PLA2G7 (0.60) ALDH1A1SLC22A12PLA2G7LMNAHTT
SCHEMBL14561810 0.80 BACE1 (0.54) ALDH1A1KDM4ELMNAHTTSMN1; SMN2
SCHEMBL12017964 0.80 SMN1; SMN2 (0.67) ALDH1A1LMNAHTTSMN1; SMN2KDM1A
SCHEMBL1627994 0.79 SLC22A12 (0.49) ALDH1A1PGRNR3C1NR3C2AR
SCHEMBL16088704 0.78 ALDH1A1 (0.76) ALDH1A1KDM4EHTTSMN1; SMN2MEN1
SCHEMBL2129695 0.78 GRM4 (0.45) ALDH1A1PGRNR3C1NR3C2AR
SCHEMBL6857747 0.78 PGR (0.52) ALDH1A1PGRNR3C1NR3C2AR
SCHEMBL2678340 0.78 SLC22A12 (0.62) PGRNR3C1NR3C2ARSLC22A12
SCHEMBL6153033 0.77 SLC6A4 (0.66) PGRPLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed