SCHEMBL6864231

SCHEMBL6864231

Cc1ccc(S(=O)(=O)N(Cc2ccccc2)c2ccc(C(O)C3CO3)c(C#N)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CNR2 P34972 5/20 0.45
CNR1 P21554 3/20 0.45
PTGES O14684 3/20 0.44
ALOX5 P09917 2/20 0.44
MAPT P10636 2/20 0.43
PGR P06401 1/20 0.43
ACHE P22303 1/20 0.42
NR1I2 O75469 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ESR1 P03372 1/20 0.40
MCL1 Q07820 1/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857706 0.87 NPSR1 (0.39) LMNAALDH1A1NPSR1MAPTPGR
SCHEMBL6864499 0.80 NR3C1 (0.57) NR3C1LMNAALDH1A1NPSR1CNR2
SCHEMBL6864234 0.79 NR3C1 (0.50) NR3C1LMNAALDH1A1NPSR1CNR2
SCHEMBL6865614 0.76 ALDH1A1 (0.64) NR3C1LMNAALDH1A1NPSR1CNR2
SCHEMBL6861888 0.72 PGR (0.36) NR3C1LMNAALDH1A1MAPTPGR
SCHEMBL22273579 0.70 NR3C1 (0.53) NR3C1LMNAALDH1A1CNR2CNR1
SCHEMBL22273557 0.70 MEN1 (0.54) NR3C1LMNAALDH1A1CNR2CNR1
SCHEMBL8169333 0.70 NR3C1 (0.54) NR3C1LMNAALDH1A1NPSR1CNR2
SCHEMBL8168003 0.70 ALDH1A1 (0.45) NR3C1LMNAALDH1A1NPSR1CNR2
SCHEMBL8171446 0.69 ALDH1A1 (0.44) NR3C1LMNAALDH1A1NPSR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed