SCHEMBL6867296

SCHEMBL6867296

CN(C)c1nc(N[C@H]2CC[C@@H](NC(=O)CCCc3cccs3)CC2)nc2c1CCCC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
TSHR P16473 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
HTT P42858 1/20 0.47
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
ADORA1 P30542 2/20 0.40
PARP1 P09874 1/20 0.38
MCHR1 Q99705 4/20 0.37
ADRA2A P08913 3/20 0.37
HRH1 P35367 2/20 0.37
HTR2B P41595 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
ADRA1A P35348 1/20 0.37
GLA P06280 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867305 1.00 MAPT (0.47) MAPTTSHRRAB9ASMN1; SMN2NPC1
SCHEMBL6872308 0.90 CYP3A4 (0.46) MAPTTSHRRAB9ASMN1; SMN2NPC1
SCHEMBL6872301 0.90 CYP3A4 (0.46) MAPTTSHRRAB9ASMN1; SMN2NPC1
SCHEMBL6878367 0.86 ADAM17 (0.40) RAB9ASMN1; SMN2NPC1BCHEACHE
SCHEMBL6878362 0.86 ADAM17 (0.40) RAB9ASMN1; SMN2NPC1BCHEACHE
SCHEMBL6867225 0.85 HPGD (0.40) MAPTRAB9ANPC1PARP1MCHR1
SCHEMBL6867228 0.85 HPGD (0.40) MAPTRAB9ANPC1PARP1MCHR1
SCHEMBL13793464 0.83 MCHR1 (0.56) PARP1MCHR1ADRA2AHRH1HTR2B
SCHEMBL7043623 0.82 MCHR1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL7043626 0.82 MCHR1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed