SCHEMBL6867905

SCHEMBL6867905

Cc1ccc(-c2nc3cc(C(=O)N(C)Cc4ccccc4)cc(N)n3n2)s1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.54
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPT P10636 2/20 0.42
POLB P06746 1/20 0.42
HSD17B2 P37059 5/20 0.41
PDE2A O00408 1/20 0.40
PDE10A Q9Y233 1/20 0.40
HSD17B1 P14061 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873684 0.89 ADORA2A (0.46) ADORA2AMEN1KMT2AMAPTALDH1A1
SCHEMBL6872164 0.86 ADORA2A (0.59) ADORA2AMEN1KMT2AMAPTALDH1A1
SCHEMBL6863226 0.82 ADORA2A (0.67) ADORA2AMEN1KMT2AALDH1A1HPGD
SCHEMBL6863351 0.81 PLAU (0.47) ADORA2AMEN1KMT2AMAPTPOLB
SCHEMBL6869917 0.81 ADORA2A (0.58) ADORA2AMEN1KMT2AALDH1A1
SCHEMBL6872068 0.81 ADORA2A (0.52) ADORA2AMEN1KMT2AALDH1A1HPGD
SCHEMBL6871437 0.81 ADORA2A (0.47) ADORA2AALDH1A1HPGD
SCHEMBL6870566 0.80 ADORA2A (0.45) ADORA2AMEN1KMT2AMAPTHSD17B2
SCHEMBL6870537 0.80 ADORA2A (0.62) ADORA2AHSD17B2HSD17B1
SCHEMBL6870638 0.80 ADORA2A (0.55) ADORA2AMEN1KMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed