SCHEMBL6863351

SCHEMBL6863351

Cc1ccc(-c2nc3cc(C(=O)NCc4ccccc4)cc(N)n3n2)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CHRM4 P08173 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863086 0.89 PLAU (0.44) PLAUHPGDKDM4EALDH1A1HSD17B10
SCHEMBL6867499 0.87 KMT2A (0.43) ALDH1A1CYP2D6HDAC3HDAC1HDAC2
SCHEMBL6870466 0.87 TP53 (0.47) HPGDKDM4EALDH1A1HSD17B10CYP2C19
SCHEMBL6872062 0.85 TP53 (0.47) HPGDKDM4EALDH1A1CYP2C19CYP2D6
SCHEMBL6869820 0.85 KDM4E (0.44) HPGDKDM4EALDH1A1HSD17B10MAPT
SCHEMBL6870449 0.85 RAB9A (0.45) PLAUHPGDALDH1A1CYP2C9HDAC3
SCHEMBL6873157 0.84 HPGDS (0.51) PLAUHPGDKDM4EALDH1A1HSD17B10
SCHEMBL6871700 0.83 SMN1; SMN2 (0.41) HPGDKDM4EALDH1A1RXFP1TP53
SCHEMBL6871437 0.81 ADORA2A (0.47) HPGDALDH1A1ADORA2A
SCHEMBL6867905 0.81 ADORA2A (0.54) HPGDALDH1A1HDAC3HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed