SCHEMBL6869675

SCHEMBL6869675

COc1ccccc1CNC(=O)c1cc(N)n2nc(-c3cccnc3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
TP53 P04637 4/20 0.51
LMNA P02545 3/20 0.49
ADORA2A P29274 1/20 0.49
HTT P42858 1/20 0.48
POLB P06746 3/20 0.48
F12 P00748 2/20 0.48
F2 P00734 2/20 0.48
MAPT P10636 2/20 0.47
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2D6 P10635 3/20 0.47
TSHR P16473 3/20 0.47
CYP2C19 P33261 3/20 0.47
HSD17B10 Q99714 3/20 0.47
CLK4 Q9HAZ1 3/20 0.47
USP2 O75604 3/20 0.47
ALOX15 P16050 2/20 0.47
MEN1 O00255 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867448 0.91 HTT (0.56) ALDH1A1TP53LMNAHTTPOLB
SCHEMBL6871512 0.87 KMT2A (0.49) ALDH1A1LMNAADORA2AF12F2
SCHEMBL6870631 0.84 LMNA (0.48) ALDH1A1TP53LMNAADORA2AHTT
SCHEMBL7114944 0.84 ADORA2A (0.54) ALDH1A1TP53LMNAADORA2AHTT
SCHEMBL6863761 0.82 HPGD (0.46) ALDH1A1TP53LMNAHTTPOLB
SCHEMBL6863441 0.82 HPGD (0.45) ALDH1A1TP53LMNAHTTPOLB
SCHEMBL6872062 0.81 TP53 (0.47) ALDH1A1TP53LMNAHTTPOLB
SCHEMBL6873996 0.81 ADORA2A (0.55) ALDH1A1TP53LMNAADORA2AHTT
SCHEMBL6871570 0.81 HPGD (0.46) ALDH1A1TP53LMNAHTTPOLB
SCHEMBL6871380 0.80 MAPT (0.46) ALDH1A1TP53LMNAADORA2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed