SCHEMBL6867448

SCHEMBL6867448

COc1ccccc1CNC(=O)c1cc(N)n2nc(-c3ccccc3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
TP53 P04637 3/20 0.55
LMNA P02545 1/20 0.55
MAPT P10636 4/20 0.52
HPGD P15428 4/20 0.49
GAA P10253 1/20 0.49
HDAC1 Q13547 1/20 0.49
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KDM4E B2RXH2 2/20 0.48
RCE1 Q9Y256 1/20 0.48
POLB P06746 1/20 0.47
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869675 0.91 ALDH1A1 (0.54) HTTTP53LMNAMAPTHPGD
SCHEMBL6870631 0.89 LMNA (0.48) HTTTP53LMNAMAPTHPGD
SCHEMBL7114944 0.87 ADORA2A (0.54) HTTTP53LMNAMAPTHPGD
SCHEMBL6863761 0.87 HPGD (0.46) HTTTP53LMNAMAPTHPGD
SCHEMBL6872062 0.86 TP53 (0.47) HTTTP53LMNAMAPTHPGD
SCHEMBL6871570 0.85 HPGD (0.46) HTTTP53LMNAMAPTHPGD
SCHEMBL6873996 0.85 ADORA2A (0.55) HTTTP53LMNAMAPTHPGD
SCHEMBL6863739 0.85 SMN1; SMN2 (0.54) TP53LMNAMAPTHPGDGAA
SCHEMBL6870074 0.85 KMT2A (0.48) LMNAMAPTHPGDALDH1A1MEN1
SCHEMBL6872927 0.85 TP53 (0.46) HTTTP53LMNAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed