SCHEMBL6870631

SCHEMBL6870631

COc1ccccc1CNC(=O)c1cc(N)n2nc(-c3ccoc3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.48
TP53 P04637 3/20 0.48
CYP1A2 P05177 4/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2C19 P33261 4/20 0.47
MAPT P10636 4/20 0.47
USP2 O75604 3/20 0.47
CYP2D6 P10635 3/20 0.47
TSHR P16473 3/20 0.47
CYP2C9 P11712 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
HTT P42858 1/20 0.46
ADORA2A P29274 2/20 0.45
ADORA1 P30542 2/20 0.45
ALDH1A1 P00352 4/20 0.45
ALOX15 P16050 2/20 0.45
CLK4 Q9HAZ1 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867448 0.89 HTT (0.56) LMNATP53MAPTMEN1KMT2A
SCHEMBL6863096 0.86 SMN1; SMN2 (0.43) LMNATP53CYP1A2CYP3A4CYP2C19
SCHEMBL6870707 0.86 KMT2A (0.43) LMNAMAPTKMT2AADORA2AALDH1A1
SCHEMBL6869746 0.84 PLAU (0.43) LMNACYP1A2CYP3A4CYP2C19MAPT
SCHEMBL6869675 0.84 ALDH1A1 (0.54) LMNATP53CYP1A2CYP3A4CYP2C19
SCHEMBL6873996 0.82 ADORA2A (0.55) LMNATP53MAPTHTTADORA2A
SCHEMBL7114944 0.82 ADORA2A (0.54) LMNATP53CYP1A2CYP3A4CYP2C19
SCHEMBL6863761 0.82 HPGD (0.46) LMNATP53CYP1A2CYP3A4CYP2C19
SCHEMBL6871380 0.82 MAPT (0.46) LMNATP53MAPTHTTADORA2A
SCHEMBL6872062 0.81 TP53 (0.47) LMNATP53CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed