SCHEMBL6863441

SCHEMBL6863441

COc1ccccc1CNC(=O)c1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 7/20 0.45
ALDH1A1 P00352 4/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
POLB P06746 2/20 0.44
TP53 P04637 2/20 0.44
GAA P10253 1/20 0.44
THRB P10828 1/20 0.44
HDAC1 Q13547 1/20 0.44
KDM4E B2RXH2 3/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
HTT P42858 1/20 0.43
RCE1 Q9Y256 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
LMNA P02545 1/20 0.43
RECQL P46063 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872927 0.86 TP53 (0.46) HPGDALDH1A1TSHRMAPK1POLB
SCHEMBL6870516 0.86 KDM4E (0.46) ALDH1A1MAPK1GAAKDM4EBCHE
SCHEMBL6870625 0.85 MAPK10 (0.45) ALDH1A1MAPK1TP53GAATHRB
SCHEMBL7114944 0.85 ADORA2A (0.54) HPGDALDH1A1POLBTP53GAA
SCHEMBL6867448 0.85 HTT (0.56) HPGDALDH1A1POLBTP53GAA
SCHEMBL6869924 0.84 CHRM4 (0.47) HPGDALDH1A1POLBTP53GAA
SCHEMBL6872062 0.82 TP53 (0.47) HPGDALDH1A1POLBTP53GAA
SCHEMBL6871570 0.82 HPGD (0.46) HPGDALDH1A1POLBTP53GAA
SCHEMBL6869675 0.82 ALDH1A1 (0.54) HPGDALDH1A1TSHRMAPK1POLB
SCHEMBL6863761 0.81 HPGD (0.46) HPGDALDH1A1POLBTP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed