SCHEMBL6869766

SCHEMBL6869766

OC(O)C(Cc1ccc(-c2ncccn2)cc1)C(O)O

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.53
CLK4 Q9HAZ1 1/20 0.40
AOC3 Q16853 2/20 0.36
CYP2A6 P11509 1/20 0.34
PPARG P37231 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HDAC4 P56524 2/20 0.33
MAPK1 P28482 1/20 0.33
AVPR2 P30518 1/20 0.32
OXTR P30559 1/20 0.32
AVPR1A P37288 1/20 0.32
PTPRA P18433 1/20 0.32
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19112147 0.81 ADRB2 (0.49) ADRB2CLK4AOC3CYP2A6PPARG
SCHEMBL19112149 0.78 ADRB2 (0.53) ADRB2CLK4AOC3CYP2A6PPARG
SCHEMBL10130811 0.77 ADRB2 (0.57) ADRB2CLK4MAPK1
SCHEMBL14122679 0.76 ADRB2 (0.52) ADRB2PPARGHDAC4PTPRA
SCHEMBL19112028 0.76 SRR (0.49) PPARG
SCHEMBL11834703 0.75 MMP12 (0.49) ADRB2PPARG
SCHEMBL533651 0.74 ADRB2 (0.63) ADRB2CLK4AOC3CYP2A6
SCHEMBL19112150 0.74 LOXL2 (0.57) ADRB2CYP2A6HDAC4
SCHEMBL31369650 0.73 SLC7A5 (0.61) ADRB2
SCHEMBL26966009 0.73 SLC7A5 (0.61) ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470514-B1 PSEUDO-DIPEPTIDES AS MMP INHIBITORS COMMISSARIAT L ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-07-12 EP disclosed
WO-2011023864-A1 PSEUDODIPEPTIDES AS MMP INHIBITORS COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2011-03-03 WO disclosed